Hemokinin 1 (human) ( —— )

产品货号. M30666 CAS No. 491851-53-7

COA

Datasheet

HNMR

HPLC

MSDS

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产品名称

Hemokinin 1 (human)
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

Endogenous substance P homolog that is a selective agonist at the tachykinin NK1 receptor (IC50 values are 1.8, 370 and 480 nM for NK1, NK3 and NK2 receptors respectively). Has proliferative and antiapoptotic actions on B-cells in vitro and is antihypertensive in vivo.
产品描述

Endogenous substance P homolog that is a selective agonist at the tachykinin NK1 receptor (IC50 values are 1.8, 370 and 480 nM for NK1, NK3 and NK2 receptors respectively). Has proliferative and antiapoptotic actions on B-cells in vitro and is antihypertensive in vivo.
同义词

——
通路

GPCR/G Protein
靶点

Neurokinin Receptor
受体

——
研究领域

——
适应症

——

CAS Number

491851-53-7
分子量

1185.4
分子式

C54H84N14O14S
纯度

>98% (HPLC)
溶解度

water:0.70 mg/mL
SMILES

[H]N[C@@H]([C@@H](C)O)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC1=CC=CC=C1)C(=O)NCC(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCSC)C(N)=O
化学全称

——

1. Bellucci et al (2002) Pharmacological profile of the novel mammalian tachykinin hemokinin 1. Br.J.Pharmacol. 135 266 PMID:

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